SCHEMBL6867481

SCHEMBL6867481

Nc1cc(C(=O)N(CCc2ccccc2)Cc2ccccc2)cc2nc(-c3ccc[nH]3)nn12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.51
RCE1 Q9Y256 1/20 0.42
PIN1 Q13526 1/20 0.39
LIMK1 P53667 1/20 0.38
LIMK2 P53671 1/20 0.38
CYP3A4 P08684 1/20 0.38
LPAR1 Q92633 3/20 0.37
LPAR5 Q9H1C0 3/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
MAPT P10636 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6867557 0.90 ADORA2A (0.46) ADORA2ALIMK1LIMK2GAAHPGD
SCHEMBL6869952 0.90 ADORA2A (0.52) ADORA2AMEN1KMT2AMAPTKDM4E
SCHEMBL6872977 0.81 ADORA2A (0.51) ADORA2ARCE1PIN1MEN1KMT2A
SCHEMBL6863393 0.78 ADORA2A (0.50) ADORA2ARCE1CYP3A4LPAR1LPAR5
SCHEMBL6867466 0.78 ADORA2A (0.49) ADORA2AKDM4EALDH1A1HPGD
SCHEMBL6870680 0.75 ADORA2A (0.60) ADORA2AKMT2AMAPTKDM4EALDH1A1
SCHEMBL6873020 0.73 ADORA2A (0.53) ADORA2ALIMK1LIMK2KDM4EGAA
SCHEMBL6873024 0.72 ADORA2A (0.75) ADORA2AMEN1KMT2AMAPTALDH1A1
SCHEMBL6863049 0.72 ADORA2A (0.45) ADORA2ACYP3A4MEN1KMT2AMAPT
SCHEMBL6863726 0.72 ADORA2A (0.56) ADORA2AMAPTKDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed