SCHEMBL6867466

SCHEMBL6867466

CCN(Cc1ccccc1F)C(=O)c1cc(N)n2nc(-c3ccc[nH]3)nc2c1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 10/20 0.49
TSPO P30536 1/20 0.37
CHRM5 P08912 1/20 0.34
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
KCNA5 P22460 1/20 0.33
ROCK2 O75116 1/20 0.33
ROCK1 Q13464 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6869952 0.87 ADORA2A (0.52) ADORA2AKDM4EALDH1A1HPGD
SCHEMBL6869841 0.82 ADORA2A (0.48) ADORA2ATSPOKDM4EALDH1A1HPGD
SCHEMBL6863381 0.80 ADORA2A (0.46) ADORA2ATSPOKDM4EALDH1A1HPGD
SCHEMBL6867557 0.79 ADORA2A (0.46) ADORA2AHPGD
SCHEMBL6867481 0.78 ADORA2A (0.51) ADORA2AKDM4EALDH1A1HPGD
SCHEMBL6870143 0.74 ADORA2A (0.65) ADORA2AKDM4EALDH1A1HPGD
SCHEMBL6867472 0.73 ADORA2A (0.40) ADORA2A
SCHEMBL6869437 0.72 KMT2A (0.47) ADORA2AALDH1A1
SCHEMBL6867645 0.72 POLB (0.49) KDM4EALDH1A1HPGDROCK2HSD17B10
SCHEMBL6863761 0.71 HPGD (0.46) KDM4EALDH1A1HPGDROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed