SCHEMBL6869952

SCHEMBL6869952

CCN(Cc1ccccc1)C(=O)c1cc(N)n2nc(-c3ccc[nH]3)nc2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.52
PPARG P37231 1/20 0.39
PLAT P00750 1/20 0.39
MAPT P10636 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
PARP1 P09874 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
DRD2 P14416 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6867557 0.91 ADORA2A (0.46) ADORA2AGAAHPGDPARP1HDAC1
SCHEMBL6867481 0.90 ADORA2A (0.51) ADORA2AMAPTKDM4EALDH1A1LMNA
SCHEMBL6867466 0.87 ADORA2A (0.49) ADORA2AKDM4EALDH1A1HPGD
SCHEMBL6863726 0.82 ADORA2A (0.56) ADORA2APPARGMAPTKDM4EALDH1A1
SCHEMBL6871681 0.80 ADORA2A (0.51) ADORA2AMAPTKDM4EALDH1A1LMNA
SCHEMBL6870601 0.80 ADORA2A (0.65) ADORA2AMAPTKDM4EALDH1A1LMNA
SCHEMBL6870657 0.80 ADORA2A (0.50) ADORA2APPARGMAPTKDM4EALDH1A1
SCHEMBL6872091 0.80 ADORA2A (0.82) ADORA2A
SCHEMBL6866841 0.79 ADORA2A (0.55) ADORA2AKDM4EALDH1A1LMNAHPGD
SCHEMBL6870143 0.78 ADORA2A (0.65) ADORA2AMAPTKDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed