SCHEMBL6867773

SCHEMBL6867773

CN(C)c1ccnc(NC2CCC(NC(=O)OCc3ccccc3)CC2)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.54
GAA P10253 1/20 0.54
TSHR P16473 1/20 0.52
EPHX1 P07099 1/20 0.49
SYK P43405 1/20 0.44
DPP4 P27487 3/20 0.44
DPP7 Q9UHL4 3/20 0.44
KCNH2 Q12809 1/20 0.44
ADORA2A P29274 1/20 0.43
ADORA1 P30542 1/20 0.43
MAPK8 P45983 2/20 0.43
MAPK9 P45984 2/20 0.43
MAPK10 P53779 1/20 0.43
CTSL P07711 1/20 0.43
CTSB P07858 1/20 0.43
CTSK P43235 1/20 0.43
JAK2 O60674 1/20 0.42
JAK1 P23458 1/20 0.42
TYK2 P29597 1/20 0.42
CA1 P00915 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6459705 0.88 GRIN2B (0.43) ALDH1A1GAAMAPK8MAPK9MAPK10
SCHEMBL6459707 0.88 GRIN2B (0.43) ALDH1A1GAAMAPK8MAPK9MAPK10
SCHEMBL6876646 0.86 MAPK8 (0.42) TSHRMAPK8MAPK9MAPK10ACHE
SCHEMBL6876639 0.86 MAPK8 (0.42) TSHRMAPK8MAPK9MAPK10ACHE
SCHEMBL6874044 0.85 AURKA (0.50) ALDH1A1MAPK8MAPK9MAPK10
SCHEMBL6874037 0.85 AURKA (0.50) ALDH1A1MAPK8MAPK9MAPK10
SCHEMBL28316716 0.85 ALDH1A1 (0.66) ALDH1A1GAATSHREPHX1DPP4
SCHEMBL21227854 0.85 ALDH1A1 (0.66) ALDH1A1GAATSHREPHX1DPP4
SCHEMBL6877124 0.82 EPHX2 (0.47) EPHX1MAPK8MAPK9MAPK10
SCHEMBL6877131 0.82 EPHX2 (0.47) EPHX1MAPK8MAPK9MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed