SCHEMBL6868013

SCHEMBL6868013

Nc1cc(C(=O)c2ccc(F)cc2)cc2nc(-c3nccs3)nn12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 13/20 0.42
NPC1 O15118 1/20 0.40
PKM P14618 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
TUBB4A P04350 1/20 0.39
TUBB P07437 1/20 0.39
TUBA3C P0DPH7 1/20 0.39
TUBA1B P68363 1/20 0.39
TUBA4A P68366 1/20 0.39
TUBB4B P68371 1/20 0.39
TUBB3 Q13509 1/20 0.39
TUBB2A Q13885 1/20 0.39
TUBB8 Q3ZCM7 1/20 0.39
TUBA3E Q6PEY2 1/20 0.39
TUBA1A Q71U36 1/20 0.39
TUBA1C Q9BQE3 1/20 0.39
TUBB6 Q9BUF5 1/20 0.39
TUBB2B Q9BVA1 1/20 0.39
TUBB1 Q9H4B7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6871431 0.89 ADORA2A (0.48) ADORA2AKMT2AADORA2BADORA1
SCHEMBL6873737 0.83 L3MBTL1 (0.43) ADORA2AKMT2AADORA1
SCHEMBL6863122 0.83 ADORA2A (0.45) ADORA2AADORA2BADORA1CHEK2
SCHEMBL6871731 0.79 ADORA2A (0.64) ADORA2A
SCHEMBL6872077 0.79 ADORA2A (0.42) ADORA2AKMT2AADORA2BADORA1
SCHEMBL6870494 0.77 ADORA2A (0.53) ADORA2AADORA2BADORA1
SCHEMBL6863814 0.77 ADORA2A (0.67) ADORA2A
SCHEMBL6871948 0.77 HDAC2 (0.46) ADORA2ANPC1RAB9AKMT2A
SCHEMBL6871350 0.76 ADORA2A (0.41) ADORA2AADORA2BADORA1
SCHEMBL6870030 0.76 ADORA2A (0.66) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed
US-6506772-B1 Pharmaceutically active salts thereof with activity as adenosine receptor ligands are disclosed. These compounds are the adenosine receptor. HOFFMANN-LA ROCHE INC. 2003-01-14 US disclosed