SCHEMBL6868489

SCHEMBL6868489

CN(C)c1nc(N[C@H]2CC[C@@H](CNCCCCCCc3ccccc3)CC2)nc2c1CCCC2

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ACHE P22303 11/20 0.40
BCHE P06276 5/20 0.40
DRD2 P14416 1/20 0.40
MCHR1 Q99705 4/20 0.39
ADRA2A P08913 3/20 0.39
NPY5R Q15761 1/20 0.39
APP P05067 1/20 0.37
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6877596 1.00 ACHE (0.40) ACHEBCHEDRD2MCHR1ADRA2A
SCHEMBL6868494 1.00 ACHE (0.40) ACHEBCHEDRD2MCHR1ADRA2A
SCHEMBL6877600 1.00 ACHE (0.40) ACHEBCHEDRD2MCHR1ADRA2A
SCHEMBL6876356 0.90 ACHE (0.41) ACHEBCHEMCHR1ADRA2A
SCHEMBL6876358 0.90 ACHE (0.41) ACHEBCHEMCHR1ADRA2A
SCHEMBL6872959 0.88 MCHR1 (0.40) ACHEBCHEMCHR1ADRA2ACTSS
SCHEMBL6872955 0.88 MCHR1 (0.40) ACHEBCHEMCHR1ADRA2ACTSS
SCHEMBL6880014 0.86 MCHR1 (0.41) ACHEMCHR1ADRA2ANPY5R
SCHEMBL6880020 0.86 MCHR1 (0.41) ACHEMCHR1ADRA2ANPY5R
SCHEMBL6876552 0.85 MCHR1 (0.42) MCHR1ADRA2ANPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed