SCHEMBL6868792

SCHEMBL6868792

COc1ccccc1-c1cnc(S(C)(=O)=O)nc1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MITF O75030 3/20 0.44
HTT P42858 3/20 0.44
NPSR1 Q6W5P4 3/20 0.44
KDM4E B2RXH2 2/20 0.44
HPGD P15428 2/20 0.44
LMNA P02545 2/20 0.44
STAT3 P40763 1/20 0.44
NPC1 O15118 6/20 0.44
RAB9A P51151 4/20 0.44
TLR9 Q9NR96 4/20 0.44
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
TP53 P04637 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
GAA P10253 1/20 0.43
SLC22A12 Q96S37 1/20 0.41
ATR Q13535 1/20 0.41
PAX8 Q06710 2/20 0.41
ALDH1A1 P00352 3/20 0.41
HSD17B10 Q99714 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6870471 0.85 NPC1 (0.43) MITFHTTNPSR1KDM4EHPGD
SCHEMBL6866170 0.83 TP53 (0.42) MITFHTTNPSR1HPGDLMNA
SCHEMBL6866618 0.83 MAPT (0.49) MITFHTTNPSR1HPGDLMNA
SCHEMBL6016467 0.81 PDE4B (0.46) MITFHTTNPSR1KDM4EHPGD
SCHEMBL6861984 0.81 MAPT (0.43) MITFHTTNPSR1KDM4EHPGD
SCHEMBL6870676 0.81 MAPT (0.42) MITFHTTNPSR1KDM4EHPGD
SCHEMBL6866602 0.78 MEN1 (0.50) KDM4EHPGDLMNANPC1KMT2A
SCHEMBL6870474 0.78 NPC1 (0.44) MITFHTTNPSR1KDM4EHPGD
SCHEMBL6871433 0.75 PTGS2 (0.44) MITFHTTNPSR1KDM4ELMNA
SCHEMBL6862136 0.74 NPC1 (0.52) MITFHTTNPSR1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1187814-B1 5-PHENYL-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2004-08-18 EP disclosed
US-6756380-B1 NEUROKININ 1 RECEPTOR ANTAGONISTS HOFFMANN-LA ROCHE INC. 2004-06-29 US disclosed
EP-1187814-A2 5-PHENYL-PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-03-20 EP disclosed
WO-2000073278-A2 5-PHENYL-PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-12-07 WO disclosed