SCHEMBL7143076

SCHEMBL7143076

CC1CCCN(C(=O)c2cc(N)n3nc(-c4ccccn4)nc3c2)C1

nearest known ligand 0.78

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 14/20 0.78
RECQL P46063 1/20 0.49
TP53 P04637 1/20 0.44
MAPT P10636 1/20 0.44
MAP3K12 Q12852 1/20 0.44
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
HPGD P15428 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6867372 0.88 ADORA2A (0.74) ADORA2AMAPT
SCHEMBL6867568 0.88 ADORA2A (1.00) ADORA2AHPGD
SCHEMBL6869099 0.87 ADORA2A (0.98) ADORA2AHPGD
SCHEMBL6871467 0.87 ADORA2A (0.98) ADORA2AHPGD
SCHEMBL6869091 0.87 ADORA2A (0.98) ADORA2AHPGD
SCHEMBL6867633 0.85 ADORA2A (0.69) ADORA2AHPGD
SCHEMBL6863273 0.85 ADORA2A (0.71) ADORA2AALDH1A1LMNAHPGD
SCHEMBL6867345 0.82 ADORA2A (0.63) ADORA2ARECQLALDH1A1HPGD
SCHEMBL6863643 0.82 ADORA2A (0.73) ADORA2AALDH1A1LMNAHPGD
SCHEMBL6871685 0.82 ADORA2A (0.80) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6506772-B1 Pharmaceutically active salts thereof with activity as adenosine receptor ligands are disclosed. These compounds are the adenosine receptor. HOFFMANN-LA ROCHE INC. 2003-01-14 US claimed
US-6506772-B1 Pharmaceutically active salts thereof with activity as adenosine receptor ligands are disclosed. These compounds are the adenosine receptor. HOFFMANN-LA ROCHE INC. 2003-01-14 US disclosed