SCHEMBL6869161

SCHEMBL6869161

CN(C)CC1CCCC=C1c1ccc(C(F)(F)F)cc1

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 3/20 0.37
SLC6A3 Q01959 2/20 0.37
SLC6A2 P23975 2/20 0.37
MCHR1 Q99705 5/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
CHKA P35790 1/20 0.34
GABBR2 O75899 3/20 0.33
GABBR1 Q9UBS5 3/20 0.33
TRPV1 Q8NER1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6861092 0.92 SLC6A4 (0.36) SLC6A4SLC6A3SLC6A2MCHR1LMNA
SCHEMBL6870938 0.92 SLC6A4 (0.36) SLC6A4SLC6A3SLC6A2MCHR1LMNA
SCHEMBL6861086 0.92 SLC6A4 (0.36) SLC6A4SLC6A3SLC6A2MCHR1LMNA
SCHEMBL5208920 0.81 SMN1; SMN2 (0.33) GAA
Hydrochloric Acid SCHEMBL4868815 0.80 SMN1; SMN2 (0.32) GAA
SCHEMBL4870450 0.77 TSHR (0.33) GAA
Hydrochloric Acid SCHEMBL4868298 0.76 TSHR (0.33)
SCHEMBL6297680 0.76 METAP1 (0.36) SLC6A4SLC6A2MCHR1LMNAGAA
SCHEMBL4870022 0.74 CHRNB2 (0.45)
SCHEMBL12020026 0.73 PDE4A (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1069106-B1 Dimethyl-(3-aryl-but-3-enyl) amine derivatives with analgesic activity GRUENENTHAL GMBH (DE) 2004-01-28 EP disclosed
EP-0799819-B1 1-Dimethylaminomethyl 2-phenyl cycloalk-2-ene derivatives with analgesic activity GRUENENTHAL GMBH (DE) 2002-09-11 EP disclosed
EP-1069106-A2 Dimethyl-(3-aryl-but-3-enyl) amine derivatives with analgesic activity Grünenthal GmbH (DE) 2001-01-17 EP disclosed
EP-0983994-A2 Pharmaceutically-active dimethyl-(3-aryl-but-3-enyl)-amine compounds Grünenthal GmbH (DE) 2000-03-08 EP disclosed
EP-0799819-A1 Dimethyl-(3-aryl-but-3-enyl) amine derivatives with analgesic activity Grünenthal GmbH (DE) 1997-10-08 EP disclosed