SCHEMBL6869223

SCHEMBL6869223

Nc1cc(C(=O)N2CCCC2)cc2nc(-c3cccs3)nn12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 14/20 1.00
ALDH1A1 P00352 2/20 0.46
NPC1 O15118 1/20 0.46
TP53 P04637 1/20 0.46
HPGD P15428 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
ERCC1 P07992 1/20 0.43
FEN1 P39748 1/20 0.43
ERCC4 Q92889 1/20 0.43
GAA P10253 1/20 0.42
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
GBA1 P04062 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6871217 0.99 ADORA2A (0.98) ADORA2AALDH1A1NPC1TP53HPGD
SCHEMBL7153750 0.83 ADORA2A (0.71) ADORA2AALDH1A1KDM4E
SCHEMBL6871909 0.82 ADORA2A (0.70) ADORA2AHPGDKDM4EKMT2A
SCHEMBL6868104 0.81 ADORA2A (0.72) ADORA2AALDH1A1HPGDMEN1KMT2A
SCHEMBL6867615 0.81 ADORA2A (0.69) ADORA2AHPGDKMT2A
SCHEMBL6867145 0.81 ADORA2A (0.71) ADORA2AALDH1A1NPC1HPGDRAB9A
SCHEMBL6867399 0.81 ADORA2A (0.67) ADORA2AALDH1A1NPC1HPGDRAB9A
SCHEMBL6863814 0.80 ADORA2A (0.67) ADORA2AHPGDKDM4E
SCHEMBL6869056 0.80 ADORA2A (0.66) ADORA2AHPGDKMT2A
SCHEMBL6870583 0.80 ADORA2A (0.66) ADORA2AALDH1A1NPC1TP53HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed
US-6506772-B1 Pharmaceutically active salts thereof with activity as adenosine receptor ligands are disclosed. These compounds are the adenosine receptor. HOFFMANN-LA ROCHE INC. 2003-01-14 US disclosed