SCHEMBL6870583

SCHEMBL6870583

COC(=O)c1cc(N)n2nc(-c3cccs3)nc2c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 8/20 0.66
MAPT P10636 3/20 0.46
NPC1 O15118 2/20 0.46
TP53 P04637 1/20 0.46
RAB9A P51151 1/20 0.46
ATM Q13315 1/20 0.46
ALDH1A1 P00352 2/20 0.46
HSD17B10 Q99714 1/20 0.46
KDM4E B2RXH2 3/20 0.45
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
GLA P06280 1/20 0.43
GAA P10253 1/20 0.43
HPGD P15428 1/20 0.43
ADORA3 P0DMS8 1/20 0.40
USP2 O75604 1/20 0.40
POLB P06746 1/20 0.40
CRHBP P24387 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7153750 0.85 ADORA2A (0.71) ADORA2AALDH1A1KDM4EADORA3ADORA1
SCHEMBL6868343 0.82 ADORA2A (0.45) ADORA2AMAPTNPC1RAB9AALDH1A1
SCHEMBL6871729 0.81 ADORA2A (0.62) ADORA2AMAPTNPC1RAB9AALDH1A1
SCHEMBL6863751 0.81 ADORA2A (0.62) ADORA2AMAPTNPC1TP53RAB9A
SCHEMBL6871212 0.81 ALDH1A1 (0.48) ADORA2AMAPTNPC1RAB9AALDH1A1
SCHEMBL6871503 0.81 ADORA2A (0.43) ADORA2AMAPTNPC1RAB9AALDH1A1
SCHEMBL6871970 0.81 ADORA2A (0.43) ADORA2AMAPTSMN1; SMN2HPGD
SCHEMBL6872088 0.80 MYC (0.56) ADORA2AMAPTNPC1RAB9AALDH1A1
SCHEMBL6870384 0.80 ADORA2A (0.58) ADORA2AMAPTALDH1A1KDM4ESMN1; SMN2
SCHEMBL6869223 0.80 ADORA2A (1.00) ADORA2ANPC1TP53RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed