SCHEMBL6869676

SCHEMBL6869676

C[C@]12CCC3c4ccc(NS(=O)(=O)O)cc4CCC3C1CCC2=O

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STS P08842 10/20 0.70
ABCC4 O15439 1/20 0.70
CYP2C9 P11712 1/20 0.70
ABCC1 P33527 1/20 0.70
SLCO1B1 Q9Y6L6 1/20 0.70
HSD17B1 P14061 3/20 0.70
CYP3A4 P08684 3/20 0.70
LMNA P02545 2/20 0.70
MAPT P10636 2/20 0.70
ESR1 P03372 2/20 0.70
ESR2 Q92731 2/20 0.70
CYP19A1 P11511 2/20 0.70
AKR1B10 O60218 1/20 0.70
SHBG P04278 1/20 0.70
CYP1A2 P05177 1/20 0.70
PGR P06401 1/20 0.70
SERPINA6 P08185 1/20 0.70
AR P10275 1/20 0.70
AKR1B1 P15121 1/20 0.70
NFKB1 P19838 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL712799 1.00 STS (0.70) STSABCC4CYP2C9ABCC1SLCO1B1
SCHEMBL17515290 0.93 STS (0.61) STSABCC4CYP2C9ABCC1SLCO1B1
SCHEMBL8408458 0.89 STS (0.71) STSABCC4CYP2C9ABCC1SLCO1B1
Estrone SCHEMBL22847 0.85 STS (0.91) STSABCC4CYP2C9ABCC1SLCO1B1
Estrone SCHEMBL6693553 0.85 STS (0.91) STSABCC4CYP2C9ABCC1SLCO1B1
Estrone SCHEMBL669802 0.84 STS (0.89) STSABCC4CYP2C9ABCC1SLCO1B1
Estrone SCHEMBL22551313 0.84 STS (0.89) STSABCC4CYP2C9ABCC1SLCO1B1
SCHEMBL22382721 0.84 STS (0.73) STSABCC4CYP2C9ABCC1SLCO1B1
Estrone SCHEMBL8901907 0.84 STS (0.89) STSABCC4CYP2C9ABCC1SLCO1B1
SCHEMBL27464072 0.84 STS (0.76) STSABCC4CYP2C9ABCC1SLCO1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0775155-B1 ESTRA-1,3,5(10)-TRIENE DERIVATIVES, METHODS OF PREPARING SUCH COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SCHERING AG (DE) 2004-05-06 EP claimed
EP-0775156-B1 PHARMACEUTICAL COMPOSITIONS CONTAINING ESTRA-1,3,5(10)-TRIENE DERIVATIVES JENAPHARM GMBH (DE) 2003-09-03 EP claimed
EP-0775155-B1 ESTRA-1,3,5(10)-TRIENE DERIVATIVES, METHODS OF PREPARING SUCH COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SCHERING AG (DE) 2004-05-06 EP disclosed