SCHEMBL8408458

SCHEMBL8408458

C[C@]12CC[C@@H]3c4ccc(NS(=O)(=O)C(F)(F)F)cc4CC[C@H]3[C@@H]1CCC2=O

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STS P08842 11/20 0.71
CA1 P00915 3/20 0.66
CA2 P00918 3/20 0.66
CA9 Q16790 3/20 0.66
CA5A P35218 2/20 0.66
HSD17B1 P14061 3/20 0.63
LMNA P02545 2/20 0.63
MAPT P10636 2/20 0.63
ESR1 P03372 2/20 0.63
ESR2 Q92731 2/20 0.63
CYP3A4 P08684 2/20 0.63
CYP19A1 P11511 2/20 0.63
AKR1B10 O60218 1/20 0.63
SHBG P04278 1/20 0.63
CYP1A2 P05177 1/20 0.63
PGR P06401 1/20 0.63
SERPINA6 P08185 1/20 0.63
AR P10275 1/20 0.63
AKR1B1 P15121 1/20 0.63
NFKB1 P19838 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6869676 0.89 STS (0.70) STSCA1CA2CA9CA5A
SCHEMBL712799 0.89 STS (0.70) STSCA1CA2CA9CA5A
SCHEMBL8411741 0.83 STS (1.00) STSCA1CA2CA9CA5A
SCHEMBL12054334 0.82 STS (0.77) STSCA1CA2CA9CA5A
SCHEMBL3825597 0.82 STS (0.77) STSCA1CA2CA9CA5A
SCHEMBL9613396 0.82 STS (0.77) STSCA1CA2CA9CA5A
SCHEMBL31321077 0.82 STS (0.77) STSCA1CA2CA9CA5A
Estrone SCHEMBL3825602 0.82 STS (0.81) STSCA1CA2CA9CA5A
SCHEMBL17515290 0.82 STS (0.61) STSCA1CA2CA9CA5A
SCHEMBL8408431 0.81 HSD17B1 (0.59) STSCA1CA2CA9CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5866603-A Derivatives of estra 1,3,5(10)triene-17-one, 3-amino compounds and their use DUQUESNE UNIVERSITY OF THE HOLY GHOST (US) 1999-02-02 US disclosed
US-5677292-A ESTROGEN SENSITIVE DISEASES; BREAST CANCER DUQUESNE UNIVERSITY OF THE HOLY GHOST (US) 1997-10-14 US disclosed
US-5571933-A Derivatives of estra 1,3,5(10)triene-17-one, 3-amino compounds and their use DUQUESNE UNIVERSITY OF THE HOLY GHOST (US) 1996-11-05 US disclosed