SCHEMBL6869801

SCHEMBL6869801

CC(CO)N(C)C.CC(COc1ncc(-c2cccc3ccccc23)c(C(=O)O)n1)N(C)C

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PPARG P37231 8/20 0.37
PPARA Q07869 8/20 0.37
ALOX5 P09917 1/20 0.37
SLC6A9 P48067 1/20 0.35
FDPS P14324 1/20 0.35
TOP1 P11387 1/20 0.34
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
HPGD P15428 1/20 0.34
AKR1C3 P42330 1/20 0.34
AKR1C2 P52895 1/20 0.34
TDP1 Q9NUW8 1/20 0.33
HTR2C P28335 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
PPARD Q03181 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6870727 0.88 ITGB1 (0.35) SLC6A9TOP1
SCHEMBL6868884 0.86 ATR (0.35) PPARGPPARASLC6A9KDM4EALDH1A1
SCHEMBL6869806 0.86 ACHE (0.42) PPARGPPARAALOX5SLC6A9TOP1
SCHEMBL6870397 0.81 HTR7 (0.37) SLC6A9KDM4EALDH1A1HPGDAKR1C3
SCHEMBL6862186 0.79 HTR1B (0.47) SLC6A9FDPSKDM4EALDH1A1HPGD
SCHEMBL6862444 0.78 HTR1B (0.48) SLC6A9FDPSKDM4EALDH1A1HTR2C
Dimethylaminoethanol SCHEMBL6868764 0.78 HTR1B (0.43) PPARGPPARASLC6A9FDPSKDM4E
SCHEMBL6870731 0.73 ACHE (0.44) SLC6A9TOP1ALDH1A1
SCHEMBL6870940 0.69 KDM4E (0.41) ALOX5KDM4EALDH1A1PPARD
SCHEMBL6868769 0.69 HTR1B (0.45) SLC6A9KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1187814-B1 5-PHENYL-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2004-08-18 EP disclosed
US-6756380-B1 NEUROKININ 1 RECEPTOR ANTAGONISTS HOFFMANN-LA ROCHE INC. 2004-06-29 US disclosed