SCHEMBL6869826

SCHEMBL6869826

CCOC(=O)c1ccc(-c2ccc3nc[nH]c(=O)c3c2)o1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 4/20 0.56
CLK2 P49760 3/20 0.56
CLK4 Q9HAZ1 3/20 0.56
DYRK1B Q9Y463 3/20 0.56
DYRK1A Q13627 2/20 0.56
ERN1 O75460 1/20 0.48
PARP1 P09874 2/20 0.46
ACVR1 Q04771 6/20 0.46
SLC2A1 P11166 1/20 0.45
IP6K1 Q92551 2/20 0.44
IP6K3 Q96PC2 1/20 0.44
IP6K2 Q9UHH9 1/20 0.44
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
TGFBR1 P36897 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12332351 0.79 PARP1 (0.57) PARP1ACVR1SLC2A1IP6K1IP6K3
SCHEMBL2116665 0.78 SLC2A1 (0.66) PARP1SLC2A1IP6K1KDM4EALDH1A1
SCHEMBL7976876 0.77 TGFBR1 (0.58) ERN1PARP1ACVR1SLC2A1IP6K1
SCHEMBL1675115 0.74 CLK1 (0.61) CLK1CLK2CLK4DYRK1BDYRK1A
SCHEMBL1675116 0.74 CLK4 (0.72) CLK1CLK2CLK4DYRK1BDYRK1A
SCHEMBL1179094 0.73 ERN1 (0.50) CLK1CLK2CLK4DYRK1BDYRK1A
SCHEMBL9911097 0.73 IP6K1 (0.66) PARP1ACVR1SLC2A1IP6K1IP6K3
SCHEMBL1675185 0.72 CLK4 (0.65) CLK1CLK2CLK4DYRK1BDYRK1A
SCHEMBL1675053 0.72 CLK1 (0.64) CLK1CLK2CLK4DYRK1BDYRK1A
SCHEMBL1675054 0.72 CLK4 (1.00) CLK1CLK2CLK4DYRK1BDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011041655-A1 QUINAZOLIN-4-AMINE DERIVATIVES; AND METHODS OF USE THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2011-04-07 WO disclosed