SCHEMBL6869931

SCHEMBL6869931

CC(C)N(Cc1ccccc1)C(=O)c1cc(N)n2nc(-c3ccc(Br)o3)nc2c1

nearest known ligand 0.72

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 18/20 0.72
ALDH1A1 P00352 2/20 0.46
TSHR P16473 2/20 0.46
GAA P10253 1/20 0.46
KMT2A Q03164 1/20 0.46
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6863514 0.90 ADORA2A (0.58) ADORA2A
SCHEMBL6863745 0.89 ADORA2A (0.57) ADORA2ATSHRLMNA
SCHEMBL6870021 0.89 ADORA2A (0.83) ADORA2AALDH1A1
SCHEMBL6873024 0.89 ADORA2A (0.75) ADORA2AALDH1A1KMT2ALMNA
SCHEMBL6869908 0.88 ADORA2A (0.80) ADORA2A
SCHEMBL6872091 0.87 ADORA2A (0.82) ADORA2A
SCHEMBL6870373 0.86 ADORA2A (0.54) ADORA2AALDH1A1TSHRGAAKMT2A
SCHEMBL6869273 0.85 ADORA2A (0.56) ADORA2A
SCHEMBL6867947 0.85 ADORA2A (0.74) ADORA2A
SCHEMBL6870569 0.84 ADORA2A (0.73) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed