SCHEMBL6869273

SCHEMBL6869273

CC(C)N(Cc1ccccc1)C(=O)c1cc(N)n2nc(-c3ccco3)nc2c1

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 10/20 0.56
PSMB5 P28074 3/20 0.50
F2 P00734 1/20 0.44
ADORA3 P0DMS8 1/20 0.43
ADORA1 P30542 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6870373 0.86 ADORA2A (0.54) ADORA2A
SCHEMBL6863514 0.86 ADORA2A (0.58) ADORA2A
SCHEMBL6869931 0.85 ADORA2A (0.72) ADORA2A
SCHEMBL6863745 0.85 ADORA2A (0.57) ADORA2A
SCHEMBL6863238 0.83 ADORA2A (0.47) ADORA2A
SCHEMBL6868951 0.82 ADORA2A (0.56) ADORA2AF2
SCHEMBL6873684 0.81 ADORA2A (0.46) ADORA2A
SCHEMBL6869779 0.81 ADORA2A (0.46) ADORA2A
SCHEMBL6863309 0.81 ADORA2A (0.69) ADORA2AF2ADORA3ADORA1
SCHEMBL6866915 0.80 PSMB5 (0.51) ADORA2APSMB5F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed