SCHEMBL6869951

SCHEMBL6869951

COc1ccc2c(C3=C4C=NC(c5cccc6cc(OC)ccc56)=C4C=N3)cccc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.44
CYP2A6 P11509 1/20 0.44
CYP11B1 P15538 3/20 0.43
CYP11B2 P19099 3/20 0.43
CYP2D6 P10635 2/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2B6 P20813 1/20 0.43
CYP2C19 P33261 1/20 0.43
MTNR1A P48039 2/20 0.39
MTNR1B P49286 2/20 0.39
RIPK3 Q9Y572 1/20 0.39
HDAC8 Q9BY41 1/20 0.38
SIRT2 Q8IXJ6 1/20 0.38
SIRT1 Q96EB6 1/20 0.38
SIRT3 Q9NTG7 1/20 0.38
SIRT5 Q9NXA8 1/20 0.38
RAB9A P51151 3/20 0.37
NPC1 O15118 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1041432 0.74 CYP1A2 (0.55) CYP1A2CYP2A6CYP11B1CYP11B2CYP2D6
SCHEMBL12592172 0.72 NPC1 (0.54) RAB9ANPC1KDM4EMEN1ALDH1A1
SCHEMBL18347012 0.72 CYP1A2 (0.52) CYP1A2CYP2A6CYP11B1CYP11B2CYP2D6
SCHEMBL13241165 0.72 MAOB (0.50) CYP1A2CYP2A6CYP11B1CYP11B2CYP2D6
SCHEMBL1402626 0.72 CYP1A2 (0.55) CYP1A2CYP2A6CYP2D6MTNR1AMTNR1B
SCHEMBL5255266 0.71 CYP1A2 (0.40) CYP1A2CYP2A6CYP11B1CYP11B2CYP2D6
SCHEMBL13241170 0.71 MAOB (0.56) CYP1A2CYP2A6CYP11B1CYP11B2CYP2D6
SCHEMBL29972803 0.70 CYP1A2 (0.53) CYP1A2CYP2A6CYP11B1CYP11B2CYP2D6
SCHEMBL443271 0.70 CYP1A2 (0.57) CYP1A2CYP2A6CYP2D6CYP3A4CYP2C9
SCHEMBL5510892 0.70 CYP1A2 (0.59) CYP1A2CYP2A6CYP11B1CYP11B2MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6805978-B2 COMPLEX CONTAINING DIKETOPYRROLO(3,4-C)PYRROLE COMPOUND TORAY INDUSTRIES, INC. (JP) 2004-10-19 US disclosed