SCHEMBL6870073

SCHEMBL6870073

CN1CCN(c2ccc(OC(=O)N(C)Cc3cc(C(F)(F)F)cc(C(F)(F)F)c3)c(-c3ccccc3Cl)c2)CC1

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 12/20 0.61
GPBAR1 Q8TDU6 2/20 0.40
SGMS2 Q8NHU3 2/20 0.40
CETP P11597 2/20 0.40
KCNH2 Q12809 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
ESR2 Q92731 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6872781 0.91 TACR1 (0.74) TACR1GPBAR1
SCHEMBL4131710 0.85 TACR1 (0.82) TACR1SGMS2
SCHEMBL6016586 0.82 TACR1 (0.64) TACR1
SCHEMBL6868287 0.80 TACR1 (0.63) TACR1GPBAR1
SCHEMBL5761333 0.77 TACR1 (0.56) TACR1
SCHEMBL6872159 0.76 TACR1 (0.49) TACR1GPBAR1
SCHEMBL4125271 0.76 TACR1 (1.00) TACR1SGMS2
SCHEMBL6637377 0.75 TACR1 (0.83) TACR1
SCHEMBL6862358 0.75 TACR1 (0.72) TACR1
SCHEMBL6016699 0.74 TACR1 (0.65) TACR1GPBAR1CETP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1171419-B1 BIPHENYL DERIVATIVES AS ANTAGONISTS OF THE NEUROKININE-1 RECEPTOR HOFFMANN LA ROCHE (CH) 2004-12-29 EP claimed