SCHEMBL6870495

SCHEMBL6870495

CN(C(=O)c1cc(N)n2nc(-c3nccs3)nc2c1)C1CCCCC1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.42
ADORA2A P29274 13/20 0.41
ALDH1A1 P00352 4/20 0.39
HPGD P15428 3/20 0.39
TSHR P16473 2/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ITK Q08881 1/20 0.37
MAPT P10636 2/20 0.36
MEN1 O00255 1/20 0.35
ALOX15 P16050 1/20 0.35
BLM P54132 1/20 0.35
KMT2A Q03164 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6871208 0.83 F2 (0.39) ADORA2AITK
SCHEMBL6871350 0.82 ADORA2A (0.41) ADORA2A
SCHEMBL6870319 0.81 ADORA2A (0.49) ADORA2AHPGD
SCHEMBL6867629 0.81 ADORA2A (0.41) ADORA2AHPGD
SCHEMBL6863074 0.81 ADORA2A (0.62) POLBADORA2AALDH1A1HPGDTSHR
SCHEMBL6863359 0.80 ADORA2A (0.47) ADORA2AHPGDTSHRSMN1; SMN2
SCHEMBL6863363 0.80 ADORA2A (0.47) ADORA2AHPGDTSHRSMN1; SMN2
SCHEMBL6871945 0.80 ADORA2A (0.42) POLBADORA2AALDH1A1HPGDTSHR
SCHEMBL6863389 0.80 NPC1 (0.47) POLBADORA2AHPGDNPC1RAB9A
SCHEMBL6863143 0.80 ADORA2A (0.58) ADORA2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed