SCHEMBL6863389

SCHEMBL6863389

CN(C(=O)c1cc(N)n2nc(-c3ccccc3)nc2c1)C1CCCCC1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
ADORA2A P29274 12/20 0.45
PTAFR P25105 1/20 0.43
PDE10A Q9Y233 1/20 0.43
POLB P06746 1/20 0.42
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
ALOX15 P16050 1/20 0.41
BLM P54132 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41
ADORA1 P30542 1/20 0.41
ITK Q08881 1/20 0.41
ATM Q13315 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6869813 0.86 ADORA2A (0.44) NPC1RAB9AADORA2APOLBMEN1
SCHEMBL6863074 0.86 ADORA2A (0.62) ADORA2APTAFRPOLBMEN1MAPT
SCHEMBL6869714 0.83 ADORA2A (0.43) NPC1RAB9AADORA2APTAFRPOLB
SCHEMBL6871451 0.82 ADORA2A (0.66) ADORA2A
SCHEMBL6863095 0.81 ADORA2A (0.67) ADORA2A
SCHEMBL6863742 0.81 ADORA2A (0.52) ADORA2APOLBMEN1MAPTHPGD
SCHEMBL6870495 0.80 POLB (0.42) NPC1RAB9AADORA2APOLBMEN1
SCHEMBL6868095 0.79 KDM4E (0.53) NPC1RAB9AADORA2AMEN1MAPT
SCHEMBL6870143 0.78 ADORA2A (0.65) NPC1RAB9AADORA2AMEN1MAPT
SCHEMBL6872164 0.78 ADORA2A (0.59) ADORA2AMEN1MAPTHPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed