SCHEMBL6863074

SCHEMBL6863074

CN(C(=O)c1cc(N)n2nc(-c3ccccn3)nc2c1)C1CCCCC1

nearest known ligand 0.62

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 11/20 0.62
POLB P06746 1/20 0.44
ALDH1A1 P00352 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
HPGD P15428 2/20 0.41
PTAFR P25105 1/20 0.41
MAPT P10636 1/20 0.41
ALOX15 P16050 1/20 0.41
BLM P54132 1/20 0.41
HSD17B10 Q99714 1/20 0.41
F12 P00748 2/20 0.40
KDM4E B2RXH2 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
F2 P00734 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6871379 0.88 ADORA2A (0.59) ADORA2AALDH1A1HSD17B10F12KDM4E
SCHEMBL6863389 0.86 NPC1 (0.47) ADORA2APOLBMEN1KMT2AHPGD
SCHEMBL6869915 0.83 ADORA2A (0.57) ADORA2AALDH1A1HSD17B10F12KDM4E
SCHEMBL6870369 0.81 ADORA2A (0.61) ADORA2AF12F2
SCHEMBL6870136 0.81 ADORA2A (0.61) ADORA2AF12F2
SCHEMBL6870495 0.81 POLB (0.42) ADORA2APOLBALDH1A1MEN1KMT2A
SCHEMBL6863310 0.81 ADORA2A (0.64) ADORA2AALDH1A1HPGDHSD17B10F12
SCHEMBL6868478 0.80 ADORA2A (0.64) ADORA2AALDH1A1HPGDHSD17B10F12
SCHEMBL6869714 0.80 ADORA2A (0.43) ADORA2APOLBALDH1A1MEN1KMT2A
SCHEMBL6871898 0.79 ADORA2A (0.62) ADORA2AMEN1KMT2AF12F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed