SCHEMBL6870780

SCHEMBL6870780

OC/C=C(\F)c1cc(-c2cccnc2)cs1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 12/20 0.51
DYRK1B Q9Y463 8/20 0.51
DYRK2 Q92630 1/20 0.45
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
CYP2A6 P11509 3/20 0.41
CYP3A4 P08684 2/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41
ERN1 O75460 1/20 0.40
CYP2C9 P11712 1/20 0.39
CYP2B6 P20813 1/20 0.39
CYP2C19 P33261 1/20 0.39
MARK3 P27448 1/20 0.38
HASPIN Q8TF76 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6870789 1.00 DYRK1A (0.51) DYRK1ADYRK1BDYRK2MKNK1MKNK2
SCHEMBL6870784 1.00 DYRK1A (0.51) DYRK1ADYRK1BDYRK2MKNK1MKNK2
SCHEMBL6880197 0.84 MMP12 (0.39) CYP3A4ERN1
SCHEMBL6851843 0.84 MMP12 (0.39) CYP3A4ERN1
SCHEMBL6880201 0.84 MMP12 (0.39) CYP3A4ERN1
SCHEMBL6852045 0.83 DYRK1A (0.54) DYRK1ADYRK1BDYRK2CYP2A6CYP3A4
SCHEMBL6852049 0.83 DYRK1A (0.54) DYRK1ADYRK1BDYRK2CYP2A6CYP3A4
SCHEMBL6852674 0.83 ERN1 (0.31) ERN1
SCHEMBL6852666 0.83 ERN1 (0.31) ERN1
SCHEMBL6852667 0.83 ERN1 (0.31) ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825170-B2 ERYTHROMYCIN TYPE MACROLIDE WITH A FUSED OXAZOLONE RING ORTHO-MCNEIL PHARMACEUTICAL, INC. 2004-11-30 US disclosed