SCHEMBL6880197

SCHEMBL6880197

OC/C=C(/F)c1cc(-c2ccncc2)cs1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 3/20 0.39
MMP13 P45452 2/20 0.39
MMP3 P08254 1/20 0.39
MMP9 P14780 1/20 0.39
MMP8 P22894 1/20 0.39
ALAD P13716 2/20 0.37
PRKCI P41743 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
QDPR P09417 1/20 0.33
MAPK14 Q16539 4/20 0.31
ERN1 O75460 1/20 0.31
KIF11 P52732 1/20 0.31
NOTUM Q6P988 1/20 0.31
CYP3A4 P08684 1/20 0.30
PRKACA P17612 1/20 0.30
ROCK1 Q13464 1/20 0.30
CYP17A1 P05093 2/20 0.30
CYP21A2 P08686 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6880201 1.00 MMP12 (0.39) MMP12MMP13MMP3MMP9MMP8
SCHEMBL6851843 1.00 MMP12 (0.39) MMP12MMP13MMP3MMP9MMP8
SCHEMBL6870780 0.84 DYRK1A (0.51) ERN1CYP3A4
SCHEMBL6870789 0.84 DYRK1A (0.51) ERN1CYP3A4
SCHEMBL6870784 0.84 DYRK1A (0.51) ERN1CYP3A4
SCHEMBL6851970 0.83 CYP3A4 (0.37) CYP3A4PRKACAROCK1
SCHEMBL6851975 0.83 CYP3A4 (0.37) CYP3A4PRKACAROCK1
SCHEMBL6852674 0.83 ERN1 (0.31) ALADERN1
SCHEMBL6852667 0.83 ERN1 (0.31) ALADERN1
SCHEMBL6852666 0.83 ERN1 (0.31) ALADERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825170-B2 ERYTHROMYCIN TYPE MACROLIDE WITH A FUSED OXAZOLONE RING ORTHO-MCNEIL PHARMACEUTICAL, INC. 2004-11-30 US disclosed