SCHEMBL6871963

SCHEMBL6871963

CC(C)CN(CC(C)C)C(=O)Oc1cc(N)n2nc(-c3nccs3)nc2c1

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 8/20 0.35
ADORA2B P29275 1/20 0.33
ADORA1 P30542 1/20 0.33
PDE11A Q9HCR9 1/20 0.32
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
ABL1 P00519 1/20 0.30
BCR P11274 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6869933 0.89 ADORA2A (0.41) ADORA2AADORA2BADORA1PDE11AABL1
SCHEMBL6873153 0.88 ADORA2A (0.38) ADORA2AADORA2BADORA1PDE11AABL1
SCHEMBL6867675 0.87 ADORA2A (0.33) ADORA2AADORA2BADORA1
SCHEMBL6869532 0.85 ADORA2A (0.36) ADORA2AADORA2BADORA1PDE11A
SCHEMBL6869890 0.84 ADORA2A (0.48) ADORA2AADORA2BADORA1PDE11A
SCHEMBL6870549 0.83 ADORA2A (0.36) ADORA2APDE11AABL1BCR
SCHEMBL6874251 0.83 ADORA2A (0.43) ADORA2AADORA2BADORA1PDE11A
SCHEMBL6869236 0.82 USP2 (0.38) ADORA2APDE11APOLB
SCHEMBL6870655 0.81 ADORA2A (0.33) ADORA2AADORA2BADORA1
SCHEMBL6863200 0.81 ADORA2A (0.38) ADORA2AADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP claimed