SCHEMBL6873153

SCHEMBL6873153

CCCN(CCC)C(=O)Oc1cc(N)n2nc(-c3nccs3)nc2c1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 10/20 0.38
F2 P00734 1/20 0.33
ADORA1 P30542 2/20 0.33
ADORA2B P29275 1/20 0.33
HSF1 Q00613 1/20 0.33
PDE11A Q9HCR9 1/20 0.33
HPGD P15428 2/20 0.32
TLR8 Q9NR97 1/20 0.31
ABL1 P00519 1/20 0.31
BCR P11274 1/20 0.31
CYP3A4 P08684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6869933 0.92 ADORA2A (0.41) ADORA2AADORA1ADORA2BHSF1PDE11A
SCHEMBL6874251 0.91 ADORA2A (0.43) ADORA2AADORA1ADORA2BHSF1PDE11A
SCHEMBL6863200 0.88 ADORA2A (0.38) ADORA2AADORA1ADORA2BHSF1HPGD
SCHEMBL6871963 0.88 ADORA2A (0.35) ADORA2AADORA1ADORA2BPDE11AABL1
SCHEMBL6869532 0.87 ADORA2A (0.36) ADORA2AADORA1ADORA2BHSF1PDE11A
SCHEMBL6869236 0.85 USP2 (0.38) ADORA2AF2PDE11A
SCHEMBL6870549 0.84 ADORA2A (0.36) ADORA2APDE11AHPGDABL1BCR
SCHEMBL6867673 0.84 ADORA2A (0.48) ADORA2AF2ADORA1ADORA2BHSF1
SCHEMBL6867675 0.83 ADORA2A (0.33) ADORA2AADORA1ADORA2B
SCHEMBL6863403 0.82 ADORA2A (0.36) ADORA2AADORA1ADORA2BHSF1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP claimed