SCHEMBL6873013

SCHEMBL6873013

Nc1cc(C(=O)NCc2ccc(F)cc2)cc2nc(-c3ccc(Cl)o3)nn12

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 12/20 0.45
L3MBTL1 Q9Y468 2/20 0.41
TP53 P04637 2/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
KMT2A Q03164 1/20 0.40
ADORA1 P30542 2/20 0.40
ADORA3 P0DMS8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6872923 0.92 ADORA2A (0.46) ADORA2ALMNAKMT2AADORA1ADORA3
SCHEMBL6871404 0.90 ADORA2A (0.51) ADORA2ATP53
SCHEMBL6871192 0.89 ADORA2A (0.58) ADORA2AL3MBTL1TP53MEN1LMNA
SCHEMBL6871992 0.83 ADORA2A (0.58) ADORA2AMEN1LMNAKMT2AADORA1
SCHEMBL6870664 0.83 TP53 (0.45) ADORA2ATP53LMNAKMT2AADORA1
SCHEMBL6871407 0.81 ADORA2A (0.48) ADORA2ALMNAKMT2A
SCHEMBL6871380 0.81 MAPT (0.46) ADORA2ATP53LMNAADORA1ADORA3
SCHEMBL6871283 0.80 PTGER2 (0.44) ADORA2AL3MBTL1TP53MEN1LMNA
SCHEMBL6863733 0.79 ADORA2A (0.50) ADORA2AMEN1KMT2A
SCHEMBL6871493 0.79 ADORA2A (0.66) ADORA2AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed