SCHEMBL6870664

SCHEMBL6870664

Nc1cc(C(=O)NCc2ccccc2Cl)cc2nc(-c3ccc(Cl)o3)nn12

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.45
ADORA2A P29274 11/20 0.45
ALDH1A1 P00352 3/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
LMNA P02545 1/20 0.44
HPGD P15428 1/20 0.44
HTT P42858 1/20 0.44
HSD17B10 Q99714 1/20 0.44
ADORA1 P30542 2/20 0.43
ADORA3 P0DMS8 1/20 0.43
ADORA2B P29275 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
GAA P10253 1/20 0.43
TSHR P16473 1/20 0.43
CYP2C19 P33261 1/20 0.43
KMT2A Q03164 1/20 0.43
MAPT P10636 1/20 0.42
ROCK2 O75116 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6871407 0.91 ADORA2A (0.48) ADORA2AALDH1A1LMNAKMT2A
SCHEMBL6871404 0.89 ADORA2A (0.51) TP53ADORA2AALDH1A1SMN1; SMN2HPGD
SCHEMBL6871380 0.88 MAPT (0.46) TP53ADORA2AALDH1A1LMNAHPGD
SCHEMBL6872375 0.87 ADORA2A (0.60) TP53ADORA2ASMN1; SMN2ADORA1ADORA3
SCHEMBL6863739 0.85 SMN1; SMN2 (0.54) TP53ALDH1A1SMN1; SMN2LMNAHPGD
SCHEMBL6872923 0.85 ADORA2A (0.46) ADORA2AALDH1A1SMN1; SMN2LMNAADORA1
SCHEMBL6871216 0.84 ADORA2A (0.44) TP53ADORA2AALDH1A1SMN1; SMN2LMNA
SCHEMBL6873013 0.83 ADORA2A (0.45) TP53ADORA2ALMNAADORA1ADORA3
SCHEMBL6868276 0.83 TP53 (0.44) TP53ADORA2AALDH1A1SMN1; SMN2LMNA
SCHEMBL6863096 0.82 SMN1; SMN2 (0.43) TP53ADORA2AALDH1A1SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed
US-6506772-B1 Pharmaceutically active salts thereof with activity as adenosine receptor ligands are disclosed. These compounds are the adenosine receptor. HOFFMANN-LA ROCHE INC. 2003-01-14 US disclosed