SCHEMBL6873199

SCHEMBL6873199

CN(C)c1nc(NC2CCC(NC(=O)NCCc3ccccc3)CC2)nc2c1CCCC2

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 4/20 0.53
NPC1 O15118 2/20 0.53
RAB9A P51151 2/20 0.53
TP53 P04637 1/20 0.53
TSHR P16473 1/20 0.53
EPHX2 P34913 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
MCHR1 Q99705 13/20 0.45
ADRA2A P08913 12/20 0.45
OPRM1 P35372 2/20 0.44
OPRL1 P41146 2/20 0.44
HRH1 P35367 2/20 0.43
HTR2B P41595 2/20 0.43
HTR1A P08908 1/20 0.43
ADRA1A P35348 1/20 0.43
NPY5R Q15761 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6873195 1.00 EPHX1 (0.53) EPHX1NPC1RAB9ATP53TSHR
SCHEMBL6875033 0.91 EPHX1 (0.51) EPHX1NPC1RAB9ASMN1; SMN2MCHR1
SCHEMBL6875039 0.91 EPHX1 (0.51) EPHX1NPC1RAB9ASMN1; SMN2MCHR1
SCHEMBL6868863 0.89 KMT2A (0.56) NPC1RAB9ASMN1; SMN2MCHR1ADRA2A
SCHEMBL6868868 0.89 KMT2A (0.56) NPC1RAB9ASMN1; SMN2MCHR1ADRA2A
SCHEMBL6831523 0.87 MCHR1 (0.45) MCHR1ADRA2AHRH1HTR2BHTR1A
SCHEMBL6831524 0.87 MCHR1 (0.45) MCHR1ADRA2AHRH1HTR2BHTR1A
SCHEMBL7043626 0.87 MCHR1 (0.44) EPHX1EPHX2MCHR1ADRA2AHRH1
SCHEMBL7043623 0.87 MCHR1 (0.44) EPHX1EPHX2MCHR1ADRA2AHRH1
SCHEMBL6878362 0.86 ADAM17 (0.40) NPC1RAB9AEPHX2SMN1; SMN2MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed