SCHEMBL6875018

SCHEMBL6875018

COc1cc(CNC[C@H]2CC[C@@H](Nc3nccc(N(C)C)n3)CC2)cc(OC)c1O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 4/20 0.43
BACE1 P56817 2/20 0.43
MCHR1 Q99705 7/20 0.39
ADRA2A P08913 2/20 0.39
NPY5R Q15761 1/20 0.39
MEN1 O00255 1/20 0.38
GAA P10253 1/20 0.38
KMT2A Q03164 1/20 0.38
DRD2 P14416 2/20 0.37
DRD3 P35462 1/20 0.37
MELK Q14680 3/20 0.36
CNR1 P21554 1/20 0.36
KCNH2 Q12809 1/20 0.36
AURKB Q96GD4 1/20 0.36
APP P05067 1/20 0.36
BCHE P06276 1/20 0.36
MAPK8 P45983 1/20 0.35
MAPK9 P45984 1/20 0.35
MAPK10 P53779 1/20 0.35
ADRA1A P35348 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6875044 1.00 ACHE (0.43) ACHEBACE1MCHR1ADRA2ANPY5R
SCHEMBL6877759 0.95 MCHR1 (0.42) ACHEBACE1MCHR1ADRA2ANPY5R
SCHEMBL6877765 0.95 MCHR1 (0.42) ACHEBACE1MCHR1ADRA2ANPY5R
SCHEMBL6457489 0.94 ACHE (0.40) ACHEBACE1MCHR1ADRA2ANPY5R
SCHEMBL6457478 0.94 ACHE (0.40) ACHEBACE1MCHR1ADRA2ANPY5R
SCHEMBL6873495 0.92 ACHE (0.51) ACHEBACE1MCHR1ADRA2ANPY5R
SCHEMBL6873488 0.92 ACHE (0.51) ACHEBACE1MCHR1ADRA2ANPY5R
SCHEMBL6467019 0.90 ACHE (0.51) ACHEBACE1MCHR1ADRA2ANPY5R
SCHEMBL6875258 0.90 ACHE (0.51) ACHEBACE1MCHR1ADRA2ANPY5R
SCHEMBL6867477 0.89 ACHE (0.44) ACHEBACE1MCHR1MEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed