SCHEMBL687539

SCHEMBL687539

Cc1ccc([C@H](CC(=O)O)NC(=O)Nc2c(O)ccn(Cc3ccccc3S(=O)(=O)N(C)C)c2=O)cc1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.36
CTSA P10619 8/20 0.35
CYP26A1 O43174 3/20 0.35
ATM Q13315 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PTGER3 P43115 1/20 0.34
MEN1 O00255 1/20 0.34
POLB P06746 1/20 0.34
KMT2A Q03164 1/20 0.34
ITGB1 P05556 2/20 0.32
ITGA4 P13612 2/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL688854 0.91 PPARG (0.39) CTSACYP26A1ATML3MBTL1PTGER3
SCHEMBL687280 0.86 POLB (0.43) CTSACYP26A1PTGER3MEN1POLB
SCHEMBL688295 0.85 MEN1 (0.39) PTGDR2CYP26A1MEN1POLBKMT2A
SCHEMBL688191 0.85 ALDH1A1 (0.40) CTSACYP26A1PTGER3MEN1POLB
SCHEMBL688155 0.85 PTGER3 (0.49) CTSAPTGER3MEN1POLBKMT2A
SCHEMBL687761 0.85 CTSA (0.46) CTSAPTGER3MEN1KMT2AALDH1A1
SCHEMBL688040 0.85 PTGER3 (0.49) CTSAPTGER3MEN1POLBKMT2A
SCHEMBL688110 0.84 MEN1 (0.49) CTSACYP26A1MEN1POLBKMT2A
SCHEMBL687559 0.83 ALDH1A1 (0.49) CTSAPTGER3POLBALDH1A1
SCHEMBL688296 0.83 CTSA (0.37) CTSACYP26A1PTGER3MEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed