SCHEMBL687559

SCHEMBL687559

COc1ccccc1Cn1ccc(O)c(NC(=O)N[C@@H](CC(=O)O)c2ccc(C)cc2)c1=O

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.49
LMNA P02545 3/20 0.47
CTSA P10619 13/20 0.45
POLB P06746 1/20 0.39
PTGER3 P43115 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL688598 0.91 ALDH1A1 (0.39) ALDH1A1LMNACTSAPOLBPTGER3
SCHEMBL687335 0.90 CTSA (0.43) CTSAPOLB
SCHEMBL687809 0.90 ITGB1 (0.39) ALDH1A1LMNACTSA
SCHEMBL687280 0.89 POLB (0.43) LMNACTSAPOLBPTGER3
SCHEMBL687449 0.88 CTSA (0.47) CTSAPOLB
SCHEMBL688191 0.88 ALDH1A1 (0.40) ALDH1A1CTSAPOLBPTGER3
SCHEMBL688040 0.88 PTGER3 (0.49) ALDH1A1CTSAPOLBPTGER3
SCHEMBL687761 0.88 CTSA (0.46) ALDH1A1LMNACTSAPTGER3
SCHEMBL688155 0.88 PTGER3 (0.49) ALDH1A1CTSAPOLBPTGER3
SCHEMBL688356 0.88 CTSA (0.45) ALDH1A1CTSAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed