SCHEMBL6875598

SCHEMBL6875598

CCOC(=O)[C@H](CC(C)C)NC(=O)NC1CCC(Nc2nc3c(c(N(C)C)n2)CCCC3)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.40
NPR3 P17342 1/20 0.40
CYP2C19 P33261 1/20 0.40
PPID Q08752 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
MCHR1 Q99705 11/20 0.36
ADRA2A P08913 8/20 0.36
HRH1 P35367 4/20 0.36
HTR2B P41595 4/20 0.36
USP2 O75604 1/20 0.35
GAA P10253 1/20 0.35
ALOX15 P16050 1/20 0.35
ADRA1A P35348 2/20 0.35
MAPK8 P45983 1/20 0.34
MAPK9 P45984 1/20 0.34
MAPK10 P53779 1/20 0.34
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
CNR1 P21554 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6875589 1.00 CYP2C9 (0.40) CYP2C9NPR3CYP2C19PPIDSMN1; SMN2
SCHEMBL6875594 1.00 CYP2C9 (0.40) CYP2C9NPR3CYP2C19PPIDSMN1; SMN2
SCHEMBL6458993 0.90 MCHR1 (0.40) CYP2C9NPR3CYP2C19PPIDSMN1; SMN2
SCHEMBL6459003 0.90 MCHR1 (0.40) CYP2C9NPR3CYP2C19PPIDSMN1; SMN2
SCHEMBL6458998 0.90 MCHR1 (0.40) CYP2C9NPR3CYP2C19PPIDSMN1; SMN2
SCHEMBL6877392 0.86 L3MBTL1 (0.41) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6877397 0.86 L3MBTL1 (0.41) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6874610 0.84 MAPK8 (0.45) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6874615 0.84 MAPK8 (0.45) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL5527235 0.81 MCHR1 (0.55) MCHR1ADRA2AHRH1HTR2BADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed