SCHEMBL6876889

SCHEMBL6876889

CN(C)C(=O)N(C)C.Nc1cc(C(=O)O)cn2nc(-c3cccs3)nc12

nearest known ligand 0.64

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 15/20 0.64
ADORA3 P0DMS8 1/20 0.38
HDAC1 Q13547 2/20 0.38
HDAC3 O15379 1/20 0.38
HDAC2 Q92769 1/20 0.38
SRPK1 Q96SB4 1/20 0.37
RPS6KB2 Q9UBS0 1/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6883012 0.83 ADORA2A (0.44) ADORA2A
SCHEMBL6886922 0.83 DHODH (0.47) ADORA2A
SCHEMBL6882930 0.82 ADORA2A (0.67) ADORA2AADORA3KDM4E
SCHEMBL6876885 0.81 ADORA2A (0.63) ADORA2AADORA3
SCHEMBL6877248 0.81 ADORA2A (0.63) ADORA2AADORA3HDAC1HDAC3HDAC2
SCHEMBL6885332 0.80 ADORA2A (0.67) ADORA2A
SCHEMBL6885020 0.80 ADORA2A (0.61) ADORA2AADORA3HDAC1HDAC3HDAC2
SCHEMBL989657 0.79 ADORA2A (0.60) ADORA2AHDAC1HDAC3HDAC2KDM4E
SCHEMBL6884914 0.78 ADORA2A (0.64) ADORA2A
SCHEMBL6887128 0.78 ADORA2A (1.00) ADORA2AHDAC1HDAC3HDAC2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6689790-B2 8-AMINO-6-AMIDO-SUBSTITUTED-(1,2,4)TRIAZOLO(1,5-A)PYRIDINES; ADENOSINE RECEPTOR MODULATERS HOFFMANN-LA ROCHE INC. 2004-02-10 US disclosed