SCHEMBL6883012

SCHEMBL6883012

CN(C)C(=O)N(C)C.Cc1ccc(-c2nc3c(N)cc(C(=O)O)cn3n2)s1

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 17/20 0.44
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
KMT2A Q03164 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6876889 0.83 ADORA2A (0.64) ADORA2A
SCHEMBL6883434 0.82 ADORA2A (0.46) ADORA2AMEN1KMT2A
SCHEMBL6886922 0.81 DHODH (0.47) ADORA2A
SCHEMBL6879225 0.81 ADORA2A (0.62) ADORA2ANPC1
SCHEMBL6876856 0.81 ADORA2A (0.64) ADORA2A
SCHEMBL6883010 0.81 ADORA2A (0.64) ADORA2A
SCHEMBL6879136 0.79 ADORA2A (0.70) ADORA2ANPC1KMT2A
SCHEMBL6884874 0.79 ADORA2A (0.67) ADORA2A
SCHEMBL6883910 0.78 ADORA2A (0.69) ADORA2AKMT2A
SCHEMBL6882517 0.78 ADORA2A (0.63) ADORA2AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6689790-B2 8-AMINO-6-AMIDO-SUBSTITUTED-(1,2,4)TRIAZOLO(1,5-A)PYRIDINES; ADENOSINE RECEPTOR MODULATERS HOFFMANN-LA ROCHE INC. 2004-02-10 US disclosed