SCHEMBL6886922

SCHEMBL6886922

CN(C)C(=O)N(C)C.Nc1cc(C(=O)O)cn2nc(-c3ccccc3)nc12

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.47
ADORA2A P29274 13/20 0.47
PARP1 P09874 1/20 0.44
GAA P10253 1/20 0.40
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
LIPE Q05469 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6884914 0.83 ADORA2A (0.64) ADORA2A
SCHEMBL6876889 0.83 ADORA2A (0.64) ADORA2A
SCHEMBL6885011 0.81 ADORA2A (0.47) DHODHADORA2APARP1GAA
SCHEMBL6883012 0.81 ADORA2A (0.44) ADORA2A
SCHEMBL6882934 0.81 ADORA2A (0.67) DHODHADORA2APARP1GAA
SCHEMBL6886917 0.81 ADORA2A (0.67) DHODHADORA2APARP1GAA
SCHEMBL989656 0.80 ADORA2A (0.70) ADORA2A
SCHEMBL6885163 0.79 ADORA2A (0.73) ADORA2A
SCHEMBL22722580 0.79 ADORA2A (0.58) DHODHADORA2APARP1GAA
SCHEMBL6887176 0.79 ADORA2A (0.60) DHODHADORA2APARP1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6689790-B2 8-AMINO-6-AMIDO-SUBSTITUTED-(1,2,4)TRIAZOLO(1,5-A)PYRIDINES; ADENOSINE RECEPTOR MODULATERS HOFFMANN-LA ROCHE INC. 2004-02-10 US disclosed