SCHEMBL687706

SCHEMBL687706

COc1cccc(F)c1Cn1cc(C)c(O)c(NC(=O)N[C@@H](CC(=O)O)c2ccc(C)cc2)c1=O

nearest known ligand 0.45

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CTSA P10619 19/20 0.45
CYP3A4 P08684 1/20 0.41
GNRHR P30968 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL688251 0.93 CTSA (0.44) CTSACYP3A4GNRHR
SCHEMBL687499 0.91 CTSA (0.45) CTSA
SCHEMBL687521 0.87 GNRHR (0.43) CTSACYP3A4GNRHR
SCHEMBL688046 0.84 CTSA (0.42) CTSACYP3A4
SCHEMBL688358 0.83 POLB (0.39) CTSACYP3A4GNRHR
SCHEMBL687715 0.83 CTSA (0.39) CTSA
SCHEMBL688604 0.83 POLB (0.41) CTSACYP3A4
SCHEMBL688871 0.83 CTSA (0.44) CTSA
SCHEMBL688146 0.83 CTSA (0.41) CTSACYP3A4
SCHEMBL688495 0.83 POLB (0.39) CTSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed