SCHEMBL688358

SCHEMBL688358

COc1cccc(Cl)c1Cn1cc(C)c(O)c(NC(=O)N[C@@H](CC(=O)O)c2ccc(C)c(C)c2)c1=O

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.39
CTSA P10619 6/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PTGER3 P43115 2/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
CYP1A2 P05177 1/20 0.35
PDE4A P27815 1/20 0.35
PDE7A Q13946 1/20 0.35
CYP3A4 P08684 2/20 0.35
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
ITGB1 P05556 2/20 0.34
ITGA4 P13612 2/20 0.34
GNRHR P30968 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL688604 0.95 POLB (0.41) POLBCTSASMN1; SMN2PTGER3MEN1
SCHEMBL687499 0.92 CTSA (0.45) POLBCTSA
SCHEMBL688220 0.91 SLC22A12 (0.36) CTSAMEN1KMT2ACYP2C9CYP2C19
SCHEMBL686879 0.91 POLB (0.36) POLBCTSASMN1; SMN2PTGER3MEN1
SCHEMBL687082 0.91 POLB (0.39) POLBCTSASMN1; SMN2MEN1KMT2A
SCHEMBL687631 0.90 SMN1; SMN2 (0.49) POLBCTSASMN1; SMN2MEN1KMT2A
SCHEMBL688501 0.90 SMN1; SMN2 (0.40) POLBCTSASMN1; SMN2PTGER3MEN1
SCHEMBL687617 0.87 POLB (0.38) POLBCTSASMN1; SMN2PTGER3MEN1
SCHEMBL688330 0.86 SMN1; SMN2 (0.40) POLBCTSASMN1; SMN2PTGER3KMT2A
SCHEMBL688170 0.86 PTGER3 (0.41) SMN1; SMN2PTGER3KDM4EALDH1A1ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed