SCHEMBL687712

SCHEMBL687712

Cc1cn(Cc2ccccc2Cl)c(=O)c(NC(=O)N[C@@H](CC(=O)O)c2cccc(OC(C)C)c2)c1O

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGER3 P43115 9/20 0.43
CNR2 P34972 1/20 0.37
SLC22A12 Q96S37 1/20 0.37
SLC16A3 O15427 1/20 0.36
SLC16A1 P53985 1/20 0.36
MCTS1 Q9ULC4 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
PPARG P37231 1/20 0.36
CTSA P10619 1/20 0.36
ITGB1 P05556 2/20 0.35
ITGA4 P13612 2/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL686799 0.93 PTGER3 (0.51) PTGER3CNR2SLC22A12SMN1; SMN2MAPT
SCHEMBL687744 0.92 PTGER3 (0.43) PTGER3CNR2SLC22A12SLC16A3SLC16A1
SCHEMBL688442 0.91 PTGER3 (0.42) PTGER3CNR2SLC22A12MAPTCTSA
SCHEMBL687045 0.91 PTGER3 (0.42) PTGER3CNR2SLC22A12MAPTCTSA
SCHEMBL688053 0.90 PTGER3 (0.43) PTGER3CNR2SLC22A12SMN1; SMN2MAPT
SCHEMBL687873 0.90 PTGER3 (0.42) PTGER3CNR2SLC22A12SLC16A3SLC16A1
SCHEMBL687348 0.89 PTGER3 (0.41) PTGER3CNR2SLC22A12SLC16A3SLC16A1
SCHEMBL688317 0.88 CNR2 (0.43) PTGER3CNR2SLC16A3SLC16A1MCTS1
SCHEMBL686846 0.88 PTGER3 (0.41) PTGER3CNR2SLC22A12SMN1; SMN2MAPT
SCHEMBL688170 0.88 PTGER3 (0.41) PTGER3CNR2SLC22A12SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed