SCHEMBL687773

SCHEMBL687773

Cc1ccc([C@H](CC(=O)O)NC(=O)Nc2c(O)c(C)cn(Cc3cc(F)ccc3Cl)c2=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CTSA P10619 18/20 0.41
PTGER3 P43115 1/20 0.37
CYP26A1 O43174 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL688871 0.93 CTSA (0.44) CTSACYP26A1
SCHEMBL688125 0.90 CTSA (0.46) CTSACYP26A1
SCHEMBL687342 0.89 CTSA (0.41) CTSAPTGER3
SCHEMBL29371834 0.88 PTGER3 (0.44) CTSAPTGER3
SCHEMBL686896 0.88 PTGER3 (0.44) CTSAPTGER3
SCHEMBL688112 0.88 KMT2A (0.41) CTSAPTGER3CYP26A1
SCHEMBL688232 0.88 CTSA (0.42) CTSACYP26A1
SCHEMBL687691 0.88 PTGER3 (0.41) CTSAPTGER3CYP26A1
SCHEMBL687893 0.87 NPSR1 (0.37) CTSAPTGER3CYP26A1
SCHEMBL688008 0.87 CTSA (0.41) CTSACYP26A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed