SCHEMBL687893

SCHEMBL687893

CCOc1ccc(Cl)c(Cn2cc(C)c(O)c(NC(=O)N[C@@H](CC(=O)O)c3ccc(C)cc3)c2=O)c1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
CTSA P10619 6/20 0.37
POLB P06746 1/20 0.36
TP53 P04637 1/20 0.35
GAA P10253 1/20 0.35
FFAR1 O14842 6/20 0.33
KEAP1 Q14145 2/20 0.33
NFE2L2 Q16236 2/20 0.33
CYP26A1 O43174 1/20 0.33
PTGER3 P43115 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL687751 0.94 SMN1; SMN2 (0.40) RXFP1CTSAPOLBGAAFFAR1
SCHEMBL687342 0.92 CTSA (0.41) NPSR1RXFP1CTSAPOLBPTGER3
SCHEMBL688112 0.92 KMT2A (0.41) CTSAPOLBKEAP1NFE2L2CYP26A1
SCHEMBL687773 0.87 CTSA (0.41) CTSACYP26A1PTGER3
SCHEMBL687744 0.86 PTGER3 (0.43) NPSR1RXFP1CTSATP53GAA
SCHEMBL29371834 0.85 PTGER3 (0.44) CTSAPTGER3
SCHEMBL686896 0.85 PTGER3 (0.44) CTSAPTGER3
SCHEMBL687640 0.85 PTGER3 (0.40) NPSR1RXFP1TP53GAAPTGER3
SCHEMBL688125 0.85 CTSA (0.46) RXFP1CTSAFFAR1CYP26A1
SCHEMBL688008 0.84 CTSA (0.41) CTSATP53GAACYP26A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed