SCHEMBL6878016

SCHEMBL6878016

CN(C)c1ccnc(N[C@H]2CC[C@@H](NC(=O)Nc3ccccc3C(F)(F)F)CC2)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 3/20 0.45
GAA P10253 1/20 0.44
TSHR P16473 2/20 0.44
ALDH1A1 P00352 1/20 0.44
CCNC P24863 2/20 0.44
CDK8 P49336 2/20 0.44
MCHR1 Q99705 3/20 0.43
ADRA2A P08913 1/20 0.43
ADRA1A P35348 1/20 0.43
HRH1 P35367 1/20 0.43
CYP3A4 P08684 2/20 0.42
P2RY1 P47900 2/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
MAPK3 P27361 4/20 0.42
CYP1A2 P05177 1/20 0.42
ALOX15 P16050 1/20 0.42
MAPK1 P28482 1/20 0.42
HIF1A Q16665 1/20 0.42
HSD17B10 Q99714 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6878023 1.00 EPHX2 (0.45) EPHX2GAATSHRALDH1A1CCNC
SCHEMBL6867232 0.91 P2RY1 (0.49) MCHR1ADRA2AADRA1AHRH1P2RY1
SCHEMBL6867237 0.91 P2RY1 (0.49) MCHR1ADRA2AADRA1AHRH1P2RY1
SCHEMBL7114626 0.89 MCHR1 (0.46) EPHX2TSHRALDH1A1MCHR1ADRA2A
SCHEMBL7114622 0.89 MCHR1 (0.46) EPHX2TSHRALDH1A1MCHR1ADRA2A
SCHEMBL6880615 0.87 CCNC (0.47) EPHX2GAACCNCCDK8MCHR1
SCHEMBL6880682 0.87 CCNC (0.44) EPHX2GAACCNCCDK8MCHR1
SCHEMBL6880688 0.87 CCNC (0.44) EPHX2GAACCNCCDK8MCHR1
SCHEMBL6880610 0.87 CCNC (0.47) EPHX2GAACCNCCDK8MCHR1
SCHEMBL6877409 0.86 KMT2A (0.56) MCHR1ADRA2AADRA1AHRH1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed