SCHEMBL6878294

SCHEMBL6878294

CCCCCC(=O)NCC1CCC(Nc2cc(N(C)C)c3ccccc3n2)CC1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.48
ALDH1A1 P00352 3/20 0.48
GAA P10253 3/20 0.48
HPGD P15428 3/20 0.48
TSHR P16473 2/20 0.48
HSD17B10 Q99714 2/20 0.48
GLA P06280 1/20 0.48
MAPK1 P28482 1/20 0.48
CNR2 P34972 6/20 0.45
CNR1 P21554 5/20 0.45
MCHR1 Q99705 3/20 0.44
EPHX2 P34913 1/20 0.42
FAAH O00519 1/20 0.41
NPY5R Q15761 2/20 0.41
ADRA2A P08913 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6878289 1.00 KDM4E (0.48) KDM4EALDH1A1GAAHPGDTSHR
SCHEMBL6876994 0.90 KDM4E (0.50) KDM4EALDH1A1GAAHPGDTSHR
SCHEMBL6877000 0.90 KDM4E (0.50) KDM4EALDH1A1GAAHPGDTSHR
SCHEMBL6878610 0.87 MCHR1 (0.48) KDM4EMCHR1NPY5RADRA2A
SCHEMBL6878604 0.87 MCHR1 (0.48) KDM4EMCHR1NPY5RADRA2A
SCHEMBL6879382 0.87 MCHR1 (0.47) KDM4EALDH1A1HPGDTSHRHSD17B10
SCHEMBL6879386 0.87 MCHR1 (0.47) KDM4EALDH1A1HPGDTSHRHSD17B10
SCHEMBL6876360 0.86 MCHR1 (0.47) KDM4EALDH1A1CNR1MCHR1EPHX2
SCHEMBL6876357 0.86 MCHR1 (0.47) KDM4EALDH1A1CNR1MCHR1EPHX2
SCHEMBL27652722 0.85 BACE1 (0.44) KDM4EALDH1A1HPGDTSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed