SCHEMBL6879382

SCHEMBL6879382

CN(C)c1cc(N[C@H]2CC[C@@H](CNC(=O)Cc3ccccc3)CC2)nc2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 2/20 0.47
ROCK2 O75116 1/20 0.43
ROCK1 Q13464 1/20 0.43
NPY5R Q15761 3/20 0.42
ADRA2A P08913 1/20 0.42
NAPEPLD Q6IQ20 3/20 0.42
ITGB3 P05106 2/20 0.41
ITGAV P06756 2/20 0.41
NPC1 O15118 2/20 0.41
KDM4E B2RXH2 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
LMNA P02545 1/20 0.41
AVPR1B P47901 1/20 0.41
ALDH1A1 P00352 3/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
RAB9A P51151 2/20 0.40
GALR3 O60755 1/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6879386 1.00 MCHR1 (0.47) MCHR1ROCK2ROCK1NPY5RADRA2A
SCHEMBL6880494 0.94 ALDH1A1 (0.48) MCHR1ROCK2ROCK1NPY5RADRA2A
SCHEMBL6873540 0.94 NPY5R (0.49) MCHR1ROCK2ROCK1NPY5RADRA2A
SCHEMBL6873544 0.94 NPY5R (0.49) MCHR1ROCK2ROCK1NPY5RADRA2A
SCHEMBL6880489 0.94 ALDH1A1 (0.48) MCHR1ROCK2ROCK1NPY5RADRA2A
SCHEMBL6876952 0.92 NPC1 (0.44) MCHR1ROCK2ROCK1NPY5RADRA2A
SCHEMBL6876960 0.92 NPC1 (0.44) MCHR1ROCK2ROCK1NPY5RADRA2A
SCHEMBL6866972 0.91 SIGMAR1 (0.44) MCHR1NPY5RADRA2ANPC1SMN1; SMN2
SCHEMBL6866974 0.91 SIGMAR1 (0.44) MCHR1NPY5RADRA2ANPC1SMN1; SMN2
SCHEMBL6872998 0.89 MCHR1 (0.51) MCHR1NPY5RADRA2AKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed