SCHEMBL6878968

SCHEMBL6878968

COC(=O)CCCCCCN(C)Cc1ccccc1

nearest known ligand 0.65

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4A O75164 2/20 0.65
KDM4C Q9H3R0 2/20 0.65
HTR7 P34969 4/20 0.59
SIGMAR1 Q99720 3/20 0.58
BCHE P06276 2/20 0.56
ACHE P22303 2/20 0.56
LTA4H P09960 1/20 0.56
APP P05067 2/20 0.54
TMEM97 Q5BJF2 1/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21908927 0.94 LTA4H (0.62) KDM4AKDM4CHTR7SIGMAR1LTA4H
SCHEMBL5522971 0.88 MEN1 (0.56) KDM4AKDM4CSIGMAR1ACHELTA4H
SCHEMBL1005793 0.87 SIGMAR1 (0.62) KDM4AKDM4CSIGMAR1LTA4HTMEM97
SCHEMBL25203501 0.87 HDAC1 (0.62) KDM4AKDM4CBCHEACHELTA4H
SCHEMBL16730590 0.87 HDAC1 (0.62) KDM4AKDM4CBCHEACHELTA4H
SCHEMBL25415046 0.86 KDM4A (0.62) KDM4AKDM4CHTR7SIGMAR1BCHE
SCHEMBL25121045 0.86 BCHE (0.74) KDM4AKDM4CSIGMAR1BCHEACHE
SCHEMBL380668 0.86 KDM4A (0.62) KDM4AKDM4CHTR7SIGMAR1BCHE
SCHEMBL7205122 0.84 KDM4A (0.76) KDM4AKDM4CHTR7SIGMAR1ACHE
SCHEMBL8904225 0.83 KDM4A (0.56) KDM4AKDM4CHTR7SIGMAR1BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200030325-A1 Reverse Amide Compounds As Protein Deacetylase Inhibitors And Methods Of Use Thereof ACETYLON PHARMACEUTICALS, INC. 2020-01-30 US disclosed
US-20170305866-A1 Histone Deacetylase 6 Selective Inhibitors for the Treatment of Bone Disease THE GENERAL HOSPITAL CORPORATION 2017-10-26 US disclosed
US-20170305866-A1 Histone Deacetylase 6 Selective Inhibitors for the Treatment of Bone Disease THE GENERAL HOSPITAL CORPORATION 2017-10-26 US disclosed
US-20160375021-A1 REVERSE AMIDE COMPOUNDS AS PROTEIN DEACETYLASE INHIBITORS AND METHODS OF USE THEREOF ACETYLON PHARMACEUTICALS, INC. 2016-12-29 US disclosed
US-9512083-B2 Histone deacetylase 6 selective inhibitors for the treatment of bone disease THE GENERAL HOSPITAL CORPORATION (US) 2016-12-06 US disclosed
US-9512083-B2 Histone deacetylase 6 selective inhibitors for the treatment of bone disease THE GENERAL HOSPITAL CORPORATION (US) 2016-12-06 US disclosed
EP-3091004-A1 REVERSE AMIDE COMPOUNDS AS PROTEIN DEACETYLASE INHIBITORS AND METHODS OF USE THEREOF Acetylon Pharmaceuticals, Inc. (US) 2016-11-09 EP disclosed
EP-2526093-B1 REVERSE AMIDE COMPOUNDS AS PROTEIN DEACETYLASE INHIBITORS AND METHODS OF USE THEREOF ACETYLON PHARMACEUTICALS INC (US) 2016-08-17 EP disclosed
US-20150045380-A1 REVERSE AMIDE COMPOUNDS AS PROTEIN DEACETYLASE INHIBITORS AND METHODS OF USE THEREOF ACETYLON PHARMACEUTICALS 2015-02-12 US disclosed
US-20150045380-A1 REVERSE AMIDE COMPOUNDS AS PROTEIN DEACETYLASE INHIBITORS AND METHODS OF USE THEREOF ACETYLON PHARMACEUTICALS 2015-02-12 US disclosed
WO-2013013113-A2 HISTONE DEACETYLASE 6 SELECTIVE INHIBITORS FOR THE TREATMENT OF BONE DISEASE THE GENERAL HOSPITAL CORPORATION (US) 2013-01-24 WO disclosed
US-20120190693-A1 Reverse Amide Compounds As Protein Deacetylase Inhibitors And Methods Of Use Thereof ACETYLON PHARMACEUTICALS, INC. 2012-07-26 US disclosed
US-20120190693-A1 Reverse Amide Compounds As Protein Deacetylase Inhibitors And Methods Of Use Thereof ACETYLON PHARMACEUTICALS, INC. 2012-07-26 US disclosed
US-20120083504-A1 Reverse Amide Compounds As Protein Deacetylase Inhibitors And Methods Of Use Thereof ACETYLON PHARMACEUTICALS, INC. 2012-04-05 US disclosed
US-20120083504-A1 Reverse Amide Compounds As Protein Deacetylase Inhibitors And Methods Of Use Thereof ACETYLON PHARMACEUTICALS, INC. 2012-04-05 US disclosed
US-8148526-B1 Reverse amide compounds as protein deacetylase inhibitors and methods of use thereof ACETYLON PHARMACEUTICALS (US) 2012-04-03 US disclosed
US-8148526-B1 Reverse amide compounds as protein deacetylase inhibitors and methods of use thereof ACETYLON PHARMACEUTICALS (US) 2012-04-03 US disclosed
US-20110300134-A1 REVERSE AMIDE COMPOUNDS AS PROTEIN DEACETYLASE INHIBITORS AND METHODS OF USE THEREOF ACETYLON PHARMACEUTICALS (US) 2011-12-08 US disclosed
US-20110300134-A1 REVERSE AMIDE COMPOUNDS AS PROTEIN DEACETYLASE INHIBITORS AND METHODS OF USE THEREOF ACETYLON PHARMACEUTICALS (US) 2011-12-08 US disclosed
WO-2011091213-A2 REVERSE AMIDE COMPOUNDS AS PROTEIN DEACETYLASE INHIBITORS AND METHODS OF USE THEREOF ACETYLON PHARMACEUTICALS (US) 2011-07-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110300134-A1 REVERSE AMIDE COMPOUNDS AS PROTEIN DEACETYLASE INHIBITORS AND METHODS OF USE THEREOF HDAC6, HDAC1, HDAC3 KDM4A 1045/4885KDM4C 2025/4885HTR7 4586/4885
US-20160375021-A1 REVERSE AMIDE COMPOUNDS AS PROTEIN DEACETYLASE INHIBITORS AND METHODS OF USE THEREOF HDAC6, HDAC1, HDAC3 KDM4A 1045/4885KDM4C 2025/4885HTR7 4586/4885
US-20150045380-A1 REVERSE AMIDE COMPOUNDS AS PROTEIN DEACETYLASE INHIBITORS AND METHODS OF USE THEREOF HDAC6, HDAC1, HDAC3 KDM4A 1045/4885KDM4C 2025/4885HTR7 4586/4885
US-20200030325-A1 Reverse Amide Compounds As Protein Deacetylase Inhibitors And Methods Of Use Thereof HDAC6, HDAC1, HDAC3 KDM4A 1045/4885KDM4C 2025/4885HTR7 4586/4885
US-20170305866-A1 Histone Deacetylase 6 Selective Inhibitors for the Treatment of Bone Disease HDAC1, HDAC6, HDAC9 KDM4A 183/4885KDM4C 412/4885HTR7 4241/4885
US-20120190693-A1 Reverse Amide Compounds As Protein Deacetylase Inhibitors And Methods Of Use Thereof HDAC6, HDAC1, HDAC3 KDM4A 1045/4885KDM4C 2025/4885HTR7 4586/4885
US-20120083504-A1 Reverse Amide Compounds As Protein Deacetylase Inhibitors And Methods Of Use Thereof HDAC6, HDAC1, HDAC3 KDM4A 1045/4885KDM4C 2025/4885HTR7 4586/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.