SCHEMBL6879682

SCHEMBL6879682

COC(=O)[C@H](CCSC)NC(=O)N[C@H]1CC[C@@H](Nc2cc(N(C)C)c3ccccc3n2)CC1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.54
LMNA P02545 1/20 0.42
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
MCHR1 Q99705 3/20 0.40
APOBEC3G Q9HC16 1/20 0.40
HTT P42858 1/20 0.40
GAA P10253 2/20 0.40
ADRA2A P08913 2/20 0.40
USP2 O75604 1/20 0.39
KMT2A Q03164 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
CASP1 P29466 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6879678 1.00 TSHR (0.54) TSHRLMNACYP3A4CYP2C19MCHR1
SCHEMBL6456529 0.87 TACR3 (0.47) TSHRMCHR1GAAADRA2A
SCHEMBL6456527 0.87 TACR3 (0.47) TSHRMCHR1GAAADRA2A
SCHEMBL4215618 0.84 MCHR1 (0.56) TSHRLMNAMCHR1ADRA2A
SCHEMBL4028824 0.84 MCHR1 (0.56) TSHRLMNAMCHR1ADRA2A
SCHEMBL4028822 0.84 MCHR1 (0.56) TSHRLMNAMCHR1ADRA2A
SCHEMBL27632422 0.81 ALDH1A1 (0.43) LMNAMCHR1ADRA2A
SCHEMBL27651737 0.81 MCHR1 (0.45) LMNAMCHR1ADRA2AKMT2A
SCHEMBL6867524 0.81 ELANE (0.44) TSHRLMNAMCHR1ADRA2A
SCHEMBL6876320 0.81 MCHR1 (0.41) MCHR1ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed