SCHEMBL6880790

SCHEMBL6880790

CN(C)c1nc(N[C@H]2CC[C@@H](NC(=S)Nc3ccccc3C(F)(F)F)CC2)nc2c1CCCC2

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.45
LMNA P02545 2/20 0.44
ALDH1A1 P00352 2/20 0.41
MAPT P10636 2/20 0.41
KDM4E B2RXH2 1/20 0.41
KDM4C Q9H3R0 1/20 0.41
MCHR1 Q99705 3/20 0.41
ADRA2A P08913 2/20 0.41
TP53 P04637 1/20 0.40
CYP2D6 P10635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6880794 1.00 PKM (0.45) PKMLMNAALDH1A1MAPTKDM4E
SCHEMBL6875875 0.89 EPHX2 (0.45) ALDH1A1MCHR1ADRA2ATP53CYP2D6
SCHEMBL6875871 0.89 EPHX2 (0.45) ALDH1A1MCHR1ADRA2ATP53CYP2D6
SCHEMBL6877751 0.88 MCHR1 (0.46) LMNAALDH1A1KDM4EMCHR1ADRA2A
SCHEMBL6877748 0.88 MCHR1 (0.46) LMNAALDH1A1KDM4EMCHR1ADRA2A
SCHEMBL6460838 0.88 MEN1 (0.40) PKMALDH1A1MAPTMCHR1ADRA2A
SCHEMBL6460846 0.88 MEN1 (0.40) PKMALDH1A1MAPTMCHR1ADRA2A
SCHEMBL6463916 0.88 MCHR1 (0.41) LMNAALDH1A1MCHR1ADRA2A
SCHEMBL6463929 0.88 MCHR1 (0.41) LMNAALDH1A1MCHR1ADRA2A
SCHEMBL6866519 0.88 GAA (0.45) LMNAALDH1A1MAPTKDM4EMCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed