SCHEMBL6875871

SCHEMBL6875871

CN(C)c1nc(N[C@H]2CC[C@@H](NC(=O)Nc3ccccc3C(F)(F)F)CC2)nc2c1CCCC2

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 4/20 0.45
MCHR1 Q99705 8/20 0.44
ADRA2A P08913 7/20 0.44
TP53 P04637 2/20 0.44
GAA P10253 1/20 0.42
ALDH1A1 P00352 2/20 0.41
TSHR P16473 1/20 0.41
POLB P06746 1/20 0.41
CYP2D6 P10635 2/20 0.41
ADRA1A P35348 2/20 0.40
HRH1 P35367 2/20 0.40
HTR2B P41595 2/20 0.40
HTR1A P08908 1/20 0.40
NPY5R Q15761 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6875875 1.00 EPHX2 (0.45) EPHX2MCHR1ADRA2ATP53GAA
SCHEMBL6874530 0.92 EPHX2 (0.56) EPHX2MCHR1ADRA2ATP53GAA
SCHEMBL6874535 0.92 EPHX2 (0.56) EPHX2MCHR1ADRA2ATP53GAA
SCHEMBL6876347 0.92 P2RY1 (0.44) MCHR1ADRA2AADRA1AHRH1HTR2B
SCHEMBL6876354 0.92 P2RY1 (0.44) MCHR1ADRA2AADRA1AHRH1HTR2B
SCHEMBL6876806 0.90 MCHR1 (0.47) EPHX2MCHR1ADRA2ATP53ALDH1A1
SCHEMBL6876812 0.90 MCHR1 (0.47) EPHX2MCHR1ADRA2ATP53ALDH1A1
SCHEMBL6880790 0.89 PKM (0.45) MCHR1ADRA2ATP53ALDH1A1CYP2D6
SCHEMBL6880794 0.89 PKM (0.45) MCHR1ADRA2ATP53ALDH1A1CYP2D6
SCHEMBL6869037 0.88 KMT2A (0.52) EPHX2MCHR1ADRA2ATP53POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed