SCHEMBL6880935

SCHEMBL6880935

COc1ccc(NC(=O)N[C@H]2CC[C@@H](Nc3cc(N(C)C)c4ccccc4n3)CC2)c(C)c1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.47
MCHR1 Q99705 1/20 0.47
SIGMAR1 Q99720 1/20 0.43
KLK7 P49862 1/20 0.43
MAPT P10636 3/20 0.43
RAB9A P51151 1/20 0.42
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
IGF1R P08069 1/20 0.41
KDR P35968 1/20 0.41
TP53 P04637 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6880943 1.00 ADRA2A (0.47) ADRA2AMCHR1SIGMAR1KLK7MAPT
SCHEMBL6880135 0.92 SIGMAR1 (0.52) ADRA2AMCHR1SIGMAR1MAPTRAB9A
SCHEMBL6880141 0.92 SIGMAR1 (0.52) ADRA2AMCHR1SIGMAR1MAPTRAB9A
SCHEMBL6874876 0.90 MCHR1 (0.43) ADRA2AMCHR1KLK7KDM4ELMNA
SCHEMBL6874884 0.90 MCHR1 (0.43) ADRA2AMCHR1KLK7KDM4ELMNA
SCHEMBL6880627 0.88 RXFP1 (0.49) ADRA2AMCHR1KDM4ELMNASMN1; SMN2
SCHEMBL6880619 0.88 RXFP1 (0.49) ADRA2AMCHR1KDM4ELMNASMN1; SMN2
SCHEMBL6466405 0.88 MCHR1 (0.46) ADRA2AMCHR1MAPTKDM4ELMNA
SCHEMBL6880443 0.88 KDR (0.51) ADRA2AMCHR1MAPTRAB9AKDM4E
SCHEMBL6880440 0.88 KDR (0.51) ADRA2AMCHR1MAPTRAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed