SCHEMBL688097

SCHEMBL688097

Cc1ccccc1NC(=O)Nc1ccc(Cn2cccc(NC(=O)N[C@@H](CC(=O)O)c3ccc4c(c3)OCO4)c2=O)cc1

nearest known ligand 0.58

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 19/20 0.58
ITGA4 P13612 19/20 0.58
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL686731 0.90 MAPT (0.55) ITGB1ITGA4RAB9A
SCHEMBL687571 0.90 ALDH1A1 (0.50) ITGB1ITGA4
SCHEMBL688325 0.88 ALDH1A1 (0.51) ITGB1ITGA4
SCHEMBL695420 0.88 MAPT (0.54) ITGB1ITGA4
SCHEMBL688223 0.86 PTGER3 (0.55) RAB9A
SCHEMBL4700630 0.85 MAPT (0.44) ITGB1ITGA4
SCHEMBL686838 0.85 PTGER3 (0.51) RAB9A
SCHEMBL687428 0.85 PTGER3 (0.56) RAB9A
SCHEMBL688073 0.85 ALDH1A1 (0.44) ITGB1ITGA4
SCHEMBL687886 0.85 PTGER3 (0.56) RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1176956-B1 CARBOXYLIC ACID DERIVATIVES THAT INHIBIT THE BINDING OF INTEGRINS TO THEIR RECEPTORS ENCYSIVE PHARMACEUTICALS INC (US) 2008-01-09 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed